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PF-04455242

PF-04455242 is a potent, selective κ-opioid receptor (KOR) antagonist with Ki of 3 nM/21 nM/22 nM for hKOR/rKOR/mKOR, respectively.

Product Specifications

CAS Number

1202647-54-8

Purity

>98%

Smiles

C1 (C2=CC=CC=C2S (N2CCCC2) (=O) =O) =CC=C (CNCC (C) C) C=C1

Molecular Formula

C21H28N2O2S

Molecular Weight

372.524224281311

Notes

For research use only.

Available Sizes

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