(R) -BAY-6035
(R) -BAY-6035 is a novel inhibitor that selectively targets the methylation of MAP3K2 by SMYD3, demonstrating nanomolar potency and specificity against kinases and other protein lysine methyltransferases.
Product Specifications
CAS Number
[2283389-29-5]
UNSPSC
12352005
Target
Histone Methyltransferase
Type
Reference compound
Related Pathways
Epigenetics
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/r-bay-6035.html
Smiles
O=C1C[C@@H](C)N(C(N2CC(C3)C3C2)=O)C4=CC=C(C(NCCC5CC5)=O)C=C4N1
Molecular Formula
C22H28N4O3
Molecular Weight
396.48
References & Citations
[1]Discovery of the SMYD3 Inhibitor BAY-6035 Using Thermal Shift Assay (TSA) -Based High-Throughput Screening
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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