TRPV1 antagonist 10
TRPV1 antagonist 10 is a potent, orally active TRPV1 antagonist with an IC50 of 33.06 nM and serves as a moderate to weak inhibitor of URAT1 (IC50 = 22.51 μM) and GLUT9 (inhibition of 60.25% at 50 μM) . It exhibits analgesic and urate-lowering properties and is applicable for research in hyperuricemia and inflammatory pain.
Product Specifications
CAS Number
896584-55-7
Field of Research
Metabolism Research, Neuroscience; Pharmacology & Drug Discovery, Pharmacology & Drug Discovery
Smiles
O=C (NC1=CC=C2OCOC2=C1) NC3=CC=C4OCCOC4=C3
Molecular Formula
C16H14N2O5
Molecular Weight
314.293
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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