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LRRK2-IN-17

LRRK2-IN-17 is an orally active LRRK2 inhibitor with IC50 values of 3.5 nM for WT and 3.3 nM for G2019S, and it also inhibits RET kinase with an IC50 of 59 nM. LRRK2-IN-17 is utilized in research related to cancer and Parkinson's disease (PD) .

Product Specifications

CAS Number

2101821-86-5

Field of Research

Cell Biology, Signal Transduction

Smiles

N (C1=C2C (=NC (NC=3N=NN (C) C3) =N1) NC=C2) [C@@H]4C=5C (CC4) =CC=CC5

Molecular Formula

C18H18N8

Molecular Weight

346.39

Storage Conditions

-20°C

Notes

For research use only.

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