ERα degrader 13
ERα degrader13 (compound MR3) is a potent ERα degrader with an IC50 of 0.55 μM. It demonstrates significant tumor regression effects in a breast cancer xenograft mouse model.
Product Specifications
CAS Number
3070968-56-5
Field of Research
Metabolism Research
Smiles
C (=O) (C1=C (SC=2C1=CC=C (O) C2) C3=CC=C (O) C=C3) C4=CC=C (OCCNC (CCCCCC/N=C/5\C=6C (C=7C (=C5) SC=8C (N7) =CC=C (N (CC) CC) C8) =CC=CC6) =O) C=C4
Molecular Formula
C50H48N4O5S2
Molecular Weight
849.07
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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