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TRPC6 antagonist-1

TRPC6 antagonist-1 (X26) is a TRPC6 inhibitor with IC50 values of 0.97 μM for TRPC6, 3.93 μM for TRPC3, 5.77 μM for TRPC5, and 4.37 μM for TRPC7. Additionally, TRPC6 antagonist-1 hinders TGF-β1-induced myofibroblast differentiation, thereby mitigating renal fibrosis.

Product Specifications

Field of Research

Neuroscience; Pharmacology & Drug Discovery, Pharmacology & Drug Discovery

Molecular Formula

C26H32N4O2S

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

Frequently Asked Questions

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