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Kv7.2/Kv7.3 activator-2

Kv7.2/Kv7.3 activator-2 is a blood-brain barrier-penetrating activator of Kv7.2/Kv7.3 channels with an EC50 of 0.25 μM. This compound exhibits excellent photostability and demonstrates potent anticonvulsant effects in acute epilepsy mouse models induced by maximal electroshock (MES) and sc-pentylenetetrazol (sc-PTZ) .

Product Specifications

Field of Research

Pharmacology & Drug Discovery

Molecular Formula

C17H20N2OS

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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