Azamulin
Azamulin is a selective, irreversible inhibitor of cytochrome P450 (CYP) 3A isoforms (IC50 values range from 26 to 240 nM for CYP3A4 and CYP3A4/5 from different sources) .It is at least 50-fold less potent against CYP2J2 and 100-fold less effective against all other CYP isoforms.Azamulin potently blocks the hydroxylation of testosterone and midazolam by CYP3A4.
Product Specifications
CAS Number
76530-44-4
Field of Research
Metabolism Research
Smiles
[H][C@@]12C (=O) CC[C@]11CC[C@@H] (C) [C@@]2 (C) [C@@H] (C[C@@] (C) (CC) [C@@H] (O) [C@@H]1C) OC (=O) CSc1nnc (N) [nH]1
Molecular Formula
C24H38N4O4S
Molecular Weight
478.65
Storage Conditions
-20°C
Notes
For research use only.
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