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GPR52 agonist-1

GPR52 agonist-1 is a potent, orally active GPR52 agonist that crosses the blood-brain barrier (pEC50:7.53) and has antipsychotic effects. GPR52 agonist-1 significantly inhibited methamphetamine-induced hyperactive behaviour in mice.

Product Specifications

CAS Number

1207965-40-9

Field of Research

Metabolism Research, Pharmacology & Drug Discovery

Smiles

O=C (NCCOC) C=1C=CC=C (C1) C2=CC=CC=3C=C (SC32) CC=4C=C (F) C=C (Cl) C4

Molecular Formula

C25H21ClFNO2S

Molecular Weight

453.96

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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