GPR52 agonist-1
GPR52 agonist-1 is a potent, orally active GPR52 agonist that crosses the blood-brain barrier (pEC50:7.53) and has antipsychotic effects. GPR52 agonist-1 significantly inhibited methamphetamine-induced hyperactive behaviour in mice.
Product Specifications
CAS Number
1207965-40-9
Field of Research
Metabolism Research, Pharmacology & Drug Discovery
Smiles
O=C (NCCOC) C=1C=CC=C (C1) C2=CC=CC=3C=C (SC32) CC=4C=C (F) C=C (Cl) C4
Molecular Formula
C25H21ClFNO2S
Molecular Weight
453.96
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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