Telcagepant
Telcagepant (MK-0974) is a small molecule CGRP receptor antagonist used in migraine research. It has been studied in vitro for receptor binding and in vivo for efficacy in preclinical migraine models, demonstrating its role in blocking CGRP-mediated neurotransmission for potential pain relief.
Product Specifications
CAS Number
781649-09-0
Product Name Alternative
MK0974, MK-0974, MK 0974, human CGRP, rhesus CGRP, Telcagepant
Field of Research
Neuroscience, Pharmacology & Drug Discovery
Purity
98.98% (May vary between batches)
Solubility
10% DMSO+40% PEG300+5% Tween 80+45% Saline:2.5 mg/mL (4.41 mM) ; DMSO:40 mg/mL (70.61 mM)
Smiles
O=C1N (C=2C (N1) =NC=CC2) C3CCN (C (N[C@H]4C (=O) N (CC (F) (F) F) C[C@@H] (CC4) C5=C (F) C (F) =CC=C5) =O) CC3
Molecular Formula
C26H27F5N6O3
Molecular Weight
566.52
Storage Conditions
-20°C
Notes
For research use only.
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
bsm-62113R-BF350-TR 20 µL
NFIB Recombinant Antibody, AbBy Fluor™ 350 Conjugated
Sign In for Pricing
View Details 