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MRS8209

MRS8209 is a selective 5-HT2B receptor antagonist (Ki = 4.27 nM) with research utility in pulmonary fibrosis. It has demonstrated protective effects on pulmonary airway opening pressure (PAO) in experimental models, supporting its application in both in vitro and in vivo studies of cardiopulmonary pathophysiology.

Product Specifications

CAS Number

3070871-46-1

Field of Research

Neuroscience, Pharmacology & Drug Discovery

Smiles

C1CCC (C1) NC2=C3C (=NC (=N2) I) N (C=N3) [C@@H]4[C@H]5C[C@]5 ([C@@H] (C4O) O) C#N

Molecular Formula

C17H19IN6O2

Molecular Weight

466.276

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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