MRS8209
MRS8209 is a selective 5-HT2B receptor antagonist (Ki = 4.27 nM) with research utility in pulmonary fibrosis. It has demonstrated protective effects on pulmonary airway opening pressure (PAO) in experimental models, supporting its application in both in vitro and in vivo studies of cardiopulmonary pathophysiology.
Product Specifications
CAS Number
3070871-46-1
Field of Research
Neuroscience, Pharmacology & Drug Discovery
Smiles
C1CCC (C1) NC2=C3C (=NC (=N2) I) N (C=N3) [C@@H]4[C@H]5C[C@]5 ([C@@H] (C4O) O) C#N
Molecular Formula
C17H19IN6O2
Molecular Weight
466.276
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog