CHI-KAT8i5
CHI-KAT8i5 is a selective KAT8 inhibitor (Kᴅ = 19.72 μM) that induces dose-dependent apoptosis. It has demonstrated antitumor activity in vitro and in vivo against various cancers, including esophageal squamous cell carcinoma, colon cancer, melanoma, gastric cancer, non-small cell lung adenocarcinoma, and liver cancer.
Product Specifications
CAS Number
2839860-29-4
Field of Research
Cell Biology, Epigenetics & Chromatin, Metabolism Research
Smiles
O=S (=O) (C=1C=CC=2N=C (SC2C1) C=CC3=CC=C (C (O) =C3) S (=O) (=O) N (CC) CC) N (CC) CC
Molecular Formula
C23H29N3O5S3
Molecular Weight
523.688
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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