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CHI-KAT8i5

CHI-KAT8i5 is a selective KAT8 inhibitor (Kᴅ = 19.72 μM) that induces dose-dependent apoptosis. It has demonstrated antitumor activity in vitro and in vivo against various cancers, including esophageal squamous cell carcinoma, colon cancer, melanoma, gastric cancer, non-small cell lung adenocarcinoma, and liver cancer.

Product Specifications

CAS Number

2839860-29-4

Field of Research

Cell Biology, Epigenetics & Chromatin, Metabolism Research

Smiles

O=S (=O) (C=1C=CC=2N=C (SC2C1) C=CC3=CC=C (C (O) =C3) S (=O) (=O) N (CC) CC) N (CC) CC

Molecular Formula

C23H29N3O5S3

Molecular Weight

523.688

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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