MOR modulator-1
MOR modulator-1 (compound 6) is a potent and selective μ opioid receptor (MOR) antagonist with Ki values of 0.25, 41.1, and 1.30 nM for μ, δ, and κ receptors, respectively. It demonstrates superior selectivity and reduced withdrawal effects compared to NAT, making it a valuable tool for in vivo behavioral studies and in vitro receptor binding assays in opioid research.
Product Specifications
CAS Number
2976336-81-7
Field of Research
Metabolism Research, Neuroscience, Pharmacology & Drug Discovery
Smiles
O[C@]12[C@@]34C=5C (O[C@]3 ([C@@H] (NC (=O) C6=NC=CS6) CC1) [H]) =C (O) C=CC5C[C@]2 (N (CC7CC7) CC4) [H]
Molecular Formula
C24H27N3O4S
Molecular Weight
453.554
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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