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ISM012-042

ISM012-042 is a potent, orally active PHD1/2 inhibitor used to study intestinal mucosal repair and immune disorders. It demonstrates protective effects on epithelial barrier integrity in vitro and exhibits anti-inflammatory activity in cell-based assays. Furthermore, it has shown efficacy in reducing inflammation and restoring barrier function in various preclinical models of experimental colitis.

Product Specifications

Field of Research

Epigenetics & Chromatin, Metabolism Research

Smiles

CC (C) (C) OC (=O) N1CCN (CC1) C2=NC3=CN=C (C (=C3C=C2) O) C (=O) NCC4=CC=C (C=C4) C#N

Molecular Formula

C26H28N6O4

Molecular Weight

488.538

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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