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CB1R antagonist 2

CB1R antagonist 2 (Compound 11g) is a selective cannabinoid receptor 1 antagonist that blocks the MAPK/NF-κB pathway, demonstrating anti-inflammatory effects in vitro by reducing LPS-induced cytokine production in RAW264.7 cells and in vivo by alleviating OVA-induced allergic rhinitis in murine models.

Product Specifications

Field of Research

Neuroscience; Pharmacology & Drug Discovery, Pharmacology & Drug Discovery, Signal Transduction

Molecular Formula

C24H26N4O

Molecular Weight

386.49

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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