CB1R antagonist 2
CB1R antagonist 2 (Compound 11g) is a selective cannabinoid receptor 1 antagonist that blocks the MAPK/NF-κB pathway, demonstrating anti-inflammatory effects in vitro by reducing LPS-induced cytokine production in RAW264.7 cells and in vivo by alleviating OVA-induced allergic rhinitis in murine models.
Product Specifications
Field of Research
Neuroscience; Pharmacology & Drug Discovery, Pharmacology & Drug Discovery, Signal Transduction
Molecular Formula
C24H26N4O
Molecular Weight
386.49
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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