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AXL/Angiokinase-IN-1

AXL/Angiokinase-IN-1 (compound 11b) is a potent, low-toxicity AXL/triple angiokinase inhibitor (IC50=3.75 nM for AXL) . It suppresses EMT and metastasis in cancer cell models (e.g., Bxpc-3, lung cancer), impairs stromal cell functions, and induces apoptosis, demonstrating utility in oncology and metastasis research.

Product Specifications

Field of Research

Cardiovascular Research, Cell Biology, Signal Transduction

Molecular Formula

C31H34ClN5O2

Molecular Weight

544.09

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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