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PDHK1-IN-1

PDHK1-IN-1 (compound 17) is a selective PDHK1 inhibitor (IC50 = 1.5 μM) that blocks phosphorylation of PDC E1α at Ser232 and Ser293, reversing PDHK1-mediated suppression of oxidative metabolism. This tool compound is used in cancer metabolism research to study the Warburg effect and has demonstrated anticancer properties in cellular assays.

Product Specifications

Field of Research

Metabolism Research

Molecular Formula

C14H11BrClNO4S

Molecular Weight

404.66

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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