ARN-6039

Product Specifications

Product Name Alternative

PF 00477736

UNSPSC Description

ARN-6039 is an orally available inverse agonist of RORγ for autoimmune demyelinating disease.

Target Antigen

ROR

Type

Reference compound

Related Pathways

Metabolic Enzyme/Protease;Vitamin D Related/Nuclear Receptor

Field of Research

Neurological Disease

Assay Protocol

https://www.medchemexpress.com/arn-6039.html

Solubility

10 mM in DMSO

Smiles

COC1=C(C=C(C2=C1)CC(C2=O)CC3=NC=CC=C3C(F)(F)F)N4CCOCC4

Molecular Weight

406.40

References & Citations

[1]Vankayalapati, Hariprasad; Yerramreddy, Venkatakrishnareddy. Preparation of dihydroindenone derivatives for use as retinoic acid-related orphan nuclear receptor modulators. US20150072980A1

Shipping Conditions

Room temperature

Product Datasheet

http://file.medchemexpress.com/batch_PDF/HY-115777/ARN-6039-DataSheet-MedChemExpress.pdf

Product MSDS

http://file.medchemexpress.com/batch_PDF/HY-115777/

Clinical Information

Phase 1

CAS Number

1675206-11-7

Available Sizes

Curated Selection

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