PI3Kδ/BET-IN-1
PI3Kδ/BET-IN-1 (compound 10b) is a potent dual inhibitor of PI3Kδ (IC50=112 nM) and BRD4-BD1 (IC50=19 nM) . It demonstrates robust antiproliferative activity in DLBCL cell models, supporting its investigation in hematological cancer research and targeted therapy development.
Product Specifications
CAS Number
3054869-10-9
Field of Research
Epigenetics & Chromatin, Signal Transduction
Smiles
O=C1C=2NC=CC2C (=CN1C) C3=NC=4C=C (SC4C (=N3) N5CCOCC5) CN6CCC (CC6) C (O) (C) C
Molecular Formula
C27H34N6O3S
Molecular Weight
522.662
Storage Conditions
-20°C
Notes
For research use only.
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