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GABAA receptor modulator-3

GABAA receptor modulator-3 (3b) acts as a positive allosteric modulator (PAM) of α1β3γ2 GABAARs, inhibiting peak and steady-state currents with IC50 values of 671 μM and 64 μM, respectively. This compound is a useful research tool for investigating GABAAR pharmacology and modulation in electrophysiological studies, both in vitro and potentially in vivo.

Product Specifications

Field of Research

Neuroscience, Pharmacology & Drug Discovery

Molecular Formula

C18H22O2

Molecular Weight

270.37

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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