GGTI-2418
GGTI-2418 is a highly potent, competitive, and selective geranylgeranyltransferase I (GGTase I) inhibitor. GGTI-2418 inhibits GGTase I and FTase activities with IC50s of 9.5 nM and 53 μM, respectively. GGTI-2418 also increases p27 (Kip1) and induces significant regression of breast tumors.
Product Specifications
CAS Number
501010-06-6
Purity
>98% (HPLC)
Solubility
In Vitro: DMSO : 125 mg/mL (283.11 mM; Ultrasonic)
Smiles
CC (C) C[C@H] (NC (=O) N1CCN (Cc2nc[nH]c2C) C (=O) [C@@H]1Cc1ccccc1) C (O) =O
Molecular Formula
C23H31N5O4
Molecular Weight
441.52
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
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