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PBRM1-BD2-IN-8

PBRM1-BD2-IN-8 (compound 34) is a potent PBRM1 Bromodomain inhibitor (PBRM1-BD2 Kd=4.4 μM, PBRM1-BD2 IC50=0.16 μM; PBRM1-BD5 Kd=25 μM) . PBRM1-BD2-IN-8 shows anti-cancer activity.

Product Specifications

CAS Number

2819989-75-6

Field of Research

Epigenetics & Chromatin

Purity

>98% (HPLC)

Solubility

In Vitro: DMSO : 100 mg/mL (315.28 mM; Ultrasonic)

Smiles

O=C1C=2C (NC (N1) C3=CC (C) =CC=C3) =CC=CC2Br

Molecular Formula

C15H13BrN2O

Molecular Weight

317.18

Storage Conditions

Storage temperature: -20°C. Stability: ≥ 2 years

Notes

For research use only.

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