WDR5-0102
WDR5-0102 is an inhibitor targeting WDR5-MLL1 interface (Kdis=7 μM, Kd=4 μM) . WDR5-0102 suppresses MLL1 HMT activity, but not human H3K4 methyltransferase SETD7 and six other HMTs: G9a, EHMT1, SUV39H2, SETD8, PRMT3, and PRMT5.
Product Specifications
CAS Number
824960-50-1
Field of Research
Epigenetics & Chromatin
Purity
>98% (HPLC)
Solubility
In Vitro: DMSO : 50 mg/mL (133.40 mM; Ultrasonic (<60°C)
Smiles
N (C (=O) C1=C (Cl) C=CC=C1) C2=C (C=CC (N (=O) =O) =C2) N3CCN (C) CC3
Molecular Formula
C18H19ClN4O3
Molecular Weight
374.82
Storage Conditions
Storage temperature: -20°C. Stability: ≥ 2 years
Notes
For research use only.
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