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Emavusertib Maleate

Emavusertib Maleate (CA-4948) is a selective IRAK4/FLT3 inhibitor with demonstrated antitumor activity in ABC DLBCL and AML models. It exhibits good oral bioavailability and has shown potent tumor growth inhibition in vivo, correlating with effective target modulation in preclinical studies.

Product Specifications

CAS Number

2376399-39-0

Field of Research

Cardiovascular Research, Cell Biology, Immunology & Inflammation, Signal Transduction

Smiles

C (=C\C (O) =O) \C (O) =O.N (C (=O) C=1N=C (OC1) C=2C=C (C) N=CC2) C3=C (N=C4C (=C3) OC (=N4) N5CCOCC5) N6CC[C@@H] (O) C6

Molecular Formula

C28H29N7O9

Molecular Weight

607.57

Storage Conditions

-20°C

Notes

For research use only.

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