SSTR4 agonist 5
Compound 5 is a potent and orally bioavailable SSTR4 agonist (EC50 = 0.228 nM) with demonstrated metabolic stability in liver microsomes. It has shown efficacy in vivo, reducing mechanical hyperalgesia in rat pain models, supporting its use in neuropharmacology and analgesic research.
Product Specifications
CAS Number
2761347-44-6
Field of Research
Pharmacology & Drug Discovery
Smiles
O=C (NC (C1=NC2=C3C (=CC=CN13) CCC2) (C) C) C4C5CNCC45C
Molecular Formula
C20H26N4O
Molecular Weight
338.447
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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