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QZ2135

QZ2135 (compound 20) is a potent and selective RET-targeting PROTAC degrader, effective against wild-type and mutant (V804M, G810C) RET fusions. It demonstrates in vivo antitumor activity in a Ba/F3-KIF5B-RET-G810C xenograft model, supporting its application in oncology research for studying RET-driven cancers and targeted protein degradation.

Product Specifications

Field of Research

Cell Biology, Pharmacology & Drug Discovery, Signal Transduction

Molecular Formula

C53H54N12O4

Molecular Weight

923.07

Storage Conditions

-20°C

Notes

For research use only.

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