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EGFR-IN-138

EGFR-IN-138 (compound 19) is a potent, small-molecule EGFR inhibitor demonstrating high potency against wild-type (IC50=37 nM), L858R mutant (IC50=2.6 nM), and T790M mutant (IC50=1.9 nM) kinases. This tool compound is suitable for in vitro biochemical and cellular assays in oncology research, particularly for studying resistance mechanisms in non-small cell lung cancer models.

Product Specifications

Field of Research

Cardiovascular Research, Cell Biology, Signal Transduction

Molecular Formula

C42H37N7O5

Molecular Weight

719.79

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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