ERα/ERβ antagonist-1
ERα/ERβ antagonist-1 (Compound 10) acts as a dual partial antagonist for both estrogen receptor subtypes, demonstrating dose-dependent inhibition of ERα and ERβ activity in HepG2 cell-based assays. This compound is a valuable research tool for investigating ER signaling in breast cancer research and endocrine system studies using in vitro models.
Product Specifications
CAS Number
2482778-93-6
Field of Research
Metabolism Research, Pharmacology & Drug Discovery
Smiles
O=C (OC1=CC=C (C=C1C=2C=CC (O) =C (C2) CC=C) CC=C) CCC
Molecular Formula
C22H24O3
Molecular Weight
336.42
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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