Melatonin-Tamoxifen Conjugate
The Melatonin-Tamoxifen Conjugate (16c) is a dual-acting small molecule that antagonizes ERα and binds melatonin MT1 receptors. It demonstrates anticancer activity in vitro, with IC50 values in the low micromolar range against breast and fibrosarcoma cell lines, and modulates β-arrestin and ERK signaling pathways.
Product Specifications
Field of Research
Pharmacology & Drug Discovery
Molecular Formula
C47H58N4O4
Molecular Weight
742.99
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
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