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TGR5 agonist 7

Compound 22-Na is a potent, orally available, and intestine-restricted TGR5 agonist (EC50 < 1 μM) . It is a valuable research tool for studying TGR5-mediated pathways in metabolic diseases, demonstrating glucose-lowering effects in murine models of diabetes.

Product Specifications

Field of Research

Pharmacology & Drug Discovery

Molecular Formula

C37H59N2NaO9S

Molecular Weight

730.93

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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