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ETP-45835 dihydrochloride

D-106669 is a cell-permeable Erk2 inhibitor with an IC50 of 18.7 μM. It potently inhibits cell proliferation with an EC50 of 0.9 μM, making it a useful tool for in vitro studies of MAPK/ERK signaling pathways in cancer and cellular growth research.

Product Specifications

CAS Number

2136571-30-5

Field of Research

Immunology & Inflammation, Signal Transduction

Smiles

C1 (C2=NNC (C3CCNCC3) =C2) =CC=NC=C1.Cl.Cl

Molecular Formula

C13H18Cl2N4

Molecular Weight

301.22

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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