MZ82
MZ82 is a potent and brain-penetrant ABCG2/BCRP inhibitor (IC50 ~23 nM), derived from Ko 143. It demonstrates superior metabolic stability in liver microsomes and improved in vivo performance in mice, making it a valuable tool for studying drug efflux and pharmacokinetics in cancer and neuroscience research.
Product Specifications
Field of Research
Pharmacology & Drug Discovery
Molecular Formula
C26H29N3O3
Molecular Weight
431.53
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
Frequently Asked Questions
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