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GPR35 activator-1

GPR35activator-1 (example 5) is a potent and selective small molecule agonist for human GPR35, demonstrating high affinity with a Ki of 0.08 nM. This compound is a valuable research tool for investigating GPR35 signaling in both in vitro cellular assays and in vivo models of metabolic and inflammatory diseases.

Product Specifications

CAS Number

2855918-34-0

Field of Research

Metabolism Research, Pharmacology & Drug Discovery, Signal Transduction

Smiles

O=C (NCC=1C=CC=CC1) C=2C=CC (=CC2) C3=CC (=CC (=C3) C4=NN=NN4) NC=5C (=O) C (=O) C5O

Molecular Formula

C25H18N6O4

Molecular Weight

466.45

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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