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PXS-4787 hydrochloride

PXS-4787 hydrochloride is a potent pan-lysyl oxidase (LOX/LOXL) inhibitor with IC50 values ranging from 0.2 to 3.2 μM across enzyme isoforms. It reduces collagen I cross-linking in human fibroblast models, supporting its use in researching fibrosis, cancer metastasis, and fibrotic disease mechanisms in vitro.

Product Specifications

CAS Number

2409964-40-3

Field of Research

Neuroscience

Smiles

S (C/C (=C/CN) /F) (=O) (=O) C1=CC=CC=C1.Cl

Molecular Formula

C10H13ClFNO2S

Molecular Weight

265.73

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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