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TLR4-IN-1

TLR4-IN-1 (compound 3k) is a potent small molecule inhibitor with an IC50 of 1.02 μM against RAW264.7 cell viability. It effectively reduces pro-inflammatory cytokine release (TNF-α, IL-1β, IL-6) in vitro and demonstrates anti-inflammatory activity in rat rheumatoid arthritis models, supporting research in immunology and inflammatory disease.

Product Specifications

CAS Number

2617578-93-3

Field of Research

Immunology & Inflammation

Smiles

O=C1C (=O) C (C) CC1C (=O) CC (=O) C

Molecular Formula

C10H12O4

Molecular Weight

196.2

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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