BI-9787
BI-9787 is a potent, zwitterionic ketohexokinase (KHK) inhibitor with IC50 values of ~12 nM against both human KHK-A and KHK-C isoforms. It demonstrates favorable metabolic stability in vitro and pharmacokinetic properties in vivo, making it a suitable tool compound for researching KHK's role in metabolic disorders such as fatty liver disease and diabetes.
Product Specifications
Molecular Formula
C24H29F2N5O2S
Molecular Weight
489.58
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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