5-HT2A/5-HT2C inverse agonist 1
This compound is a potent dual 5-HT2A/5-HT2C receptor inverse agonist with hERG-inhibiting properties, reducing cardiovascular risk. It demonstrates significant antipsychotic activity in the MK-801-induced mouse model, making it a valuable tool for in vivo psychosis research and in vitro receptor pharmacology studies.
Product Specifications
CAS Number
2718990-76-0
Field of Research
Neuroscience, Pharmacology & Drug Discovery
Smiles
N (CC1=NN (C) C=C1) (C (NCC2=CC=C (OCCC) C=C2) =O) [C@@H]3C4 (CC4) CN (C) CC3
Molecular Formula
C24H35N5O2
Molecular Weight
425.57
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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