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INOS/TopoI-IN-1

INOS/TopoI-IN-1 (AuL9) is a dual-target inhibitor of Topoisomerase I (K_i=2.72 μM) and iNOS (K_i=1.49 μM), exhibiting anti-tumor activity in vitro against breast cancer cells (MCF-7 IC50=3.5 μM; MDA-MB-231 IC50=6.3 μM) by inducing DNA damage and apoptosis.

Product Specifications

Field of Research

Cell Biology, Immunology & Inflammation, Molecular Biology, Signal Transduction

Molecular Formula

C34H40AuBrCl2N3OS

Molecular Weight

886.54

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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