INOS/TopoI-IN-1
INOS/TopoI-IN-1 (AuL9) is a dual-target inhibitor of Topoisomerase I (K_i=2.72 μM) and iNOS (K_i=1.49 μM), exhibiting anti-tumor activity in vitro against breast cancer cells (MCF-7 IC50=3.5 μM; MDA-MB-231 IC50=6.3 μM) by inducing DNA damage and apoptosis.
Product Specifications
Field of Research
Cell Biology, Immunology & Inflammation, Molecular Biology, Signal Transduction
Molecular Formula
C34H40AuBrCl2N3OS
Molecular Weight
886.54
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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