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DS03090629

DS03090629 is a potent, orally bioavailable MEK inhibitor with sub-nanomolar binding affinity for MEK and phospho-MEK. It effectively inhibits proliferation in BRAF-mutant melanoma cell lines and is a valuable research tool for studying MAPK pathway dysregulation in oncology, supporting both in vitro and in vivo preclinical investigations.

Product Specifications

Field of Research

Signal Transduction

Molecular Formula

C25H26ClN5O2

Molecular Weight

463.96

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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