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PARP1-IN-27

PARP1-IN-27 (Compound 9B) is a potent dual PARP1/2 inhibitor with low nanomolar IC50 values. It demonstrates anti-proliferative activity in BRCA-mutant cell lines by inducing DNA damage, ROS, G2/M arrest, and apoptosis, supporting its use in oncology research for studying DNA repair mechanisms and synthetic lethality.

Product Specifications

Field of Research

Cell Biology, Epigenetics & Chromatin, Immunology & Inflammation, Metabolism Research, Molecular Biology, Signal Transduction

Molecular Formula

C17H12FNO4

Molecular Weight

313.28

Storage Conditions

-20°C

Notes

For research use only.

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