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HPK1-IN-47

HPK1-IN-47 is a potent PROTAC-based degrader of HPK1 (DC50 = 23 nM in PBMCs) used as a key chemical precursor. It enables research into HPK1-mediated diseases, such as cancer, through both in vitro cellular studies and in vivo experimental models.

Product Specifications

CAS Number

2893885-42-0

Field of Research

Pharmacology & Drug Discovery, Signal Transduction

Smiles

O=C (C=1C=CC (=CC1C) C2=CNC=3N=CC (=NC32) C4=CC (=C5C (=C4) CCNC5) C) N (C) C

Molecular Formula

C26H27N5O

Molecular Weight

425.53

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

Frequently Asked Questions

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