W4275
W4275 is a potent, orally bioavailable, and selective NSD2 inhibitor (IC50 = 17 nM) . It demonstrates antiproliferative effects in RS411 cells (IC50 = 230 nM) and significantly suppresses tumor growth in RS411 xenograft models, supporting its utility in oncology research for studying epigenetic targets.
Product Specifications
CAS Number
3051650-00-8
Field of Research
Epigenetics & Chromatin
Smiles
N#CC=1N=C2C=C (OCCCN3CCOCC3) C (OC) =CC2=C (N1) NC4CCN (CC4) C (C) C
Molecular Formula
C25H36N6O3
Molecular Weight
468.59
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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