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DS06652923

DS06652923 is a potent, orally bioavailable small molecule inhibitor targeting EGFR triple mutations. It demonstrates strong in vitro activity with a GI50 of 9.4 nM in Ba/F3-EGFRdel19/T790M/C795S cells and has shown efficacy in vivo by inducing tumor regression in a syngeneic transplantation model, supporting its use in oncology research for resistant NSCLC.

Product Specifications

Field of Research

Cardiovascular Research, Signal Transduction

Storage Conditions

-20°C

Notes

For research use only.

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