GPR17 modulator-1
GPR17 Modulator-1 (Compound 2-046) is a potent, brain-penetrant small molecule antagonist of human GPR17 (IC50 < 10 nM) . Its moderate PK profile supports its use in both cellular assays and in vivo rodent models for researching neuroinflammatory and demyelinating diseases.
Product Specifications
CAS Number
3039853-91-0
Field of Research
Signal Transduction
Smiles
O=S (=O) (NC1=CC (F) =C (N=C1OC) OCC (F) F) C=2C=NN3C=C (Cl) C=CC23
Molecular Formula
C15H12ClF3N4O4S
Molecular Weight
436.79
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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