[Nle20] H4 peptide (16−23)
The [Nle20] H4 peptide (16–23) is a potent and selective SETD8 inhibitor (Kd = 0.14 μM) that acts by competing for the histone substrate binding site. This tool compound is used in epigenetic research to study histone methylation's role in cancer cell proliferation and as a lead for anticancer therapeutic development.
Product Specifications
CAS Number
2042178-19-6
Smiles
[C@H] (CC1=CN=CN1) (C (N[C@H] (C (N[C@H] (C (N[C@H] (C (N[C@H] (C (N[C@@H] (CCCNC (=N) N) C (O) =O) =O) CC (C) C) =O) C (C) C) =O) CCCC) =O) CCCNC (=N) N) =O) NC ([C@@H] (NC ([C@H] (CCCCN) N) =O) CCCNC (=N) N) =O
Molecular Formula
C47H88N20O9
Molecular Weight
1077.33
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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