Adenosine receptor antagonist 5
Compound 39 is a potent and selective human A3 adenosine receptor antagonist (Ki = 12 nM) . It inhibits IB-MECA-induced cAMP production in vitro and demonstrates anti-proliferative effects in LK-2 and NCI-H1792 cancer cell lines, while exhibiting rapid metabolism in human liver microsomes.
Product Specifications
Field of Research
Neuroscience, Pharmacology & Drug Discovery
Storage Conditions
-20°C
Notes
For research use only.
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